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Sterically controlled stereoregulations in aldol reactions of 3-aryl-1-alkyl dihydrothiouracils

Publication Type : Journal Article

Publisher : Thieme

Source : Synlett, 2011

Url : https://www.thieme-connect.com/products/ejournals/html/10.1055/s-0031-1289889

Campus : Amritapuri

School : School of Biotechnology

Verified : No

Year : 2011

Abstract : Aldol reactions of 3-aryl-1-alkyl dihydrothiouracils were investigated with respect to the orientation of the exocyclic group at N1, electronic effects of the aryl substituent at N3 and the steric demands of the electrophile. The reactions highlight the preference for formation of the anti aldol diastereomer with increasing steric constraints of the reactants.

Cite this Research Publication : Varun Kumar, Gopal L. Khatik and Vipin A. Nair, "Sterically controlled stereoregulations in aldol reactions of 3-aryl-1-alkyl dihydrothiouracils", Synlett, 2011, 22, 2997-3001.

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